Juan José
Vaquero López
Profesor/a Emérito/a


Instituto Ramón y Cajal de Investigación Sanitaria
Madrid, EspañaPublications in collaboration with researchers from Instituto Ramón y Cajal de Investigación Sanitaria (14)
2023
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One-Pot (3 + 2) Cycloaddition-Isomerization-Oxidation of 2,2,2-Trifluorodiazoethane and Styryl Derivatives
Journal of Organic Chemistry, Vol. 88, Núm. 15, pp. 11258-11262
2022
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Highly efficient unbridged D-A+(D) chromophores based on the quinolizinium cation for nonlinear optical (NLO) applications
Dyes and Pigments, Vol. 205
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Pyridazino-pyrrolo-quinoxalinium salts as highly potent and selective leishmanicidal agents targeting trypanothione reductase
European Journal of Medicinal Chemistry, Vol. 227
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RICORS2040: The need for collaborative research in chronic kidney disease
Clinical Kidney Journal, Vol. 15, Núm. 3, pp. 372-387
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Visible-Light-Mediated Regioselective Chlorosulfonylation of Acrylamides
Synthesis (Germany), Vol. 55, Núm. 11, pp. 1783-1791
2021
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A Computer-Driven Scaffold-Hopping Approach Generating New PTP1B Inhibitors from the Pyrrolo[1,2-a]quinoxaline Core
ChemMedChem, Vol. 16, Núm. 18, pp. 2895-2906
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Enantioselective Copper-Catalyzed Synthesis of Trifluoromethyl-Cyclopropylboronates
Organic Letters, Vol. 23, Núm. 15, pp. 6174-6178
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Pyrrolo[1,2-a]quinoxal-5-inium salts and 4,5-dihydropyrrolo[1,2-a]quinoxalines: Synthesis, activity and computational docking for protein tyrosine phosphatase 1B
Bioorganic and Medicinal Chemistry, Vol. 44
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Recent developments in the chemistry of BN-aromatic hydrocarbons
Advances in Heterocyclic Chemistry (Academic Press Inc.), pp. 197-259
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Tripeptides as Integrin-Linked Kinase Modulating Agents Based on a Protein-Protein Interaction with α-Parvin
ACS Medicinal Chemistry Letters, Vol. 12, Núm. 11, pp. 1656-1662
2020
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Gold-catalyzed synthetic strategies towards four-carbon ring systems
Catalysts, Vol. 10, Núm. 10, pp. 1-47
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Pyrrolo[1,2-a]quinoxalines: Insulin Mimetics that Exhibit Potent and Selective Inhibition against Protein Tyrosine Phosphatase 1B
ChemMedChem, Vol. 15, Núm. 19, pp. 1788-1801
2019
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MAP3K kinases and kidney injury
Nefrologia, Vol. 39, Núm. 6, pp. 568-580
2018
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Discovery of potent calpain inhibitors based on the azolo-imidazolidenone scaffold
European Journal of Medicinal Chemistry, Vol. 157, pp. 946-959