Diseño, interacción y síntesis de compuestos biológicamente activos - Design, interaction and synthesis of bioactive compounds.
DISCOBAC
University of Sfax
Sfax, Túnez
Publikationen in Zusammenarbeit mit Forschern von University of Sfax (10)
2025
2024
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Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors
ACS Chemical Neuroscience, Vol. 15, Núm. 18, pp. 3363-3383
2023
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Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer’s Disease Treatment
International Journal of Molecular Sciences, Vol. 24, Núm. 11
2021
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Synthesis and Biological Assessment of PyrimidoTacrines as Promising Agents for Alzheimer's Disease Therapy
ChemistrySelect, Vol. 6, Núm. 37, pp. 9975-9980
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Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments
Chemical Record, Vol. 21, Núm. 1, pp. 162-174
2020
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Triazolopyridopyrimidine: A new scaffold for dual-target small molecules for Alzheimer's disease therapy
Molecules, Vol. 25, Núm. 14
2019
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Multi-target 1,4-dihydropyridines showing calcium channel blockade and antioxidant capacity for Alzheimer's disease therapy
Bioorganic Chemistry, Vol. 91
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New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H3 Receptor (H3R) Antagonism and Calcium Channels Blockade with Additional Cholinesterase Inhibition
Journal of Medicinal Chemistry, Vol. 62, Núm. 24, pp. 11416-11422
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Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer’s disease therapy
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 34, Núm. 1, pp. 163-170
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Synthesis of (±)-cis-1-Aryl-3-oxo-2,3-dihydro-1H-benzo[f]chromene-2-carbonitriles and (±)-trans-4-Aryl-2-oxo-3,4-dihydro-2H-benzo[h]chromene-3-carbonitriles
ChemistrySelect, Vol. 4, Núm. 44, pp. 12902-12905