Diseño, interacción y síntesis de compuestos biológicamente activos - Design, interaction and synthesis of bioactive compounds.
DISCOBAC
Universidad Autónoma de Madrid
Madrid, España
2025
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Contilistat, a New Multitarget Small Polyfunctionalized Indole Derivative
Synlett, Vol. 36, Núm. 16, pp. 2655-2660
2024
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Contilisant+Tubastatin A Hybrids: Polyfunctionalized Indole Derivatives as New HDAC Inhibitor-Based Multitarget Small Molecules with In Vitro and In Vivo Activity in Neurodegenerative Diseases
Journal of Medicinal Chemistry, Vol. 67, Núm. 18, pp. 16533-16555
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Ni(2,2′:6′,2′′-terpyridine)2: a high-spin octahedral formal Ni(0) complex
Dalton Transactions, Vol. 53, Núm. 20, pp. 8550-8554
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Nickel-catalyzed cycloisomerization of 1,5-allenynes
Advanced Synthesis and Catalysis, Vol. 366, Núm. 4, pp. 790-797
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Synthesis of ladderanes by nickel-catalyzed cyclodimerization of allenynes: scope and mechanism
Advanced Synthesis and Catalysis, Vol. 366, Núm. 22, pp. 4755-4764
2023
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Metal-catalyzed borylative cyclization reactions of polyunsaturated substrates for the synthesis of heterocycles
Targets in Heterocyclic Systems, Vol. 27, pp. 309-340
2022
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Nickel-catalyzed hydroborylative polycyclization of allenynes: an atom-economical and diastereoselective synthesis of bicyclic 5-5 fused rings
Advanced Synthesis and Catalysis, Vol. 364, Núm. 10, pp. 1716-1723
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Polyfunctionalized α-Phenyl-tert-butyl(benzyl)nitrones: Multifunctional Antioxidants for Stroke Treatment
Antioxidants, Vol. 11, Núm. 9
2021
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On the mechanism of the formation of alkyl-Ni(i) catalysts
Chemical Communications, Vol. 57, Núm. 19, pp. 2424-2427
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Pd-catalyzed C(sp3)-C(sp) bond formation in iodocyclobutenes
Chemical Communications, Vol. 57, Núm. 68, pp. 8456-8459
2020
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In Vitro and in Silico ADME-Tox Profiling and Safety Significance of Multifunctional Monoamine Oxidase Inhibitors Targeting Neurodegenerative Diseases
ACS Chemical Neuroscience, Vol. 11, Núm. 22, pp. 3793-3801
2019
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Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer’s disease therapy
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 34, Núm. 1, pp. 479-489
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New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H3 Receptor (H3R) Antagonism and Calcium Channels Blockade with Additional Cholinesterase Inhibition
Journal of Medicinal Chemistry, Vol. 62, Núm. 24, pp. 11416-11422
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Quinoxalinetacrine QT78, a cholinesterase inhibitor as a potential ligand for Alzheimer’s disease therapy
Molecules, Vol. 24, Núm. 8