DISCOBAC
Diseño, interacción y síntesis de compuestos biológicamente activos ; Design, interaction and synthesis of bioactive compounds.
Publicaciones (75) Publicaciones en las que ha participado algún/a investigador/a
2024
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Contilisant+Tubastatin A Hybrids: Polyfunctionalized Indole Derivatives as New HDAC Inhibitor-Based Multitarget Small Molecules with In Vitro and In Vivo Activity in Neurodegenerative Diseases
Journal of Medicinal Chemistry, Vol. 67, Núm. 18, pp. 16533-16555
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Cs2CO3-Promoted Alkylation of 3-Cyano-2(1H)-Pyridones: Anticancer Evaluation and Molecular Docking
ChemPlusChem
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DNA Interactions and Biological Activity of 2,9-Disubstituted 1,10-Phenanthroline Thiosemicarbazone-Based Ligands and a 4-Phenylthiazole Derivative
Biology, Vol. 13, Núm. 1
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Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors
ACS Chemical Neuroscience, Vol. 15, Núm. 18, pp. 3363-3383
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Fluorescent Vitamin B12–Platinum(II) Derivatives as Potential Metallotheranostic Agents for the Treatment and Imaging of Tumors
Inorganics, Vol. 12, Núm. 3
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Ni(2,2′:6′,2′′-terpyridine)2: a high-spin octahedral formal Ni(0) complex
Dalton Transactions, Vol. 53, Núm. 20, pp. 8550-8554
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Nickel-Catalyzed Cycloisomerization of 1,5-Allenynes
Advanced Synthesis and Catalysis, Vol. 366, Núm. 4, pp. 790-797
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Synthesis, structural study and antitumor activity of novel alditol-based imidazophenanthrolines (aldo-IPs)
Bioorganic and Medicinal Chemistry, Vol. 99
2023
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Carbohydrate effect of novel arene Ru(II) phenanthroline-glycoconjugates on metastatic biological processes
Journal of Inorganic Biochemistry, Vol. 247
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Delivery of Therapeutic Biopolymers Employing Silica-Based Nanosystems
Pharmaceutics, Vol. 15, Núm. 2
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Embedded Pressure Sensing Metamaterials Using TPU-Graphene Composites and Additive Manufacturing
IEEE Sensors Journal, Vol. 23, Núm. 15, pp. 16656-16664
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Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer’s Disease Treatment
International Journal of Molecular Sciences, Vol. 24, Núm. 11
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Gold-catalyzed endo-selective cyclization of alkynylcyclobutanecarboxamides: synthesis of cyclobutane-fused dihydropyridones
Organic and Biomolecular Chemistry, Vol. 21, Núm. 13, pp. 2705-2708
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METAL-CATALYZED BORYLATIVE CYCLIZATION REACTIONS OF POLYUNSATURATED SUBSTRATES FOR THE SYNTHESIS OF HETEROCYCLES
Targets in Heterocyclic Systems, Vol. 27, pp. 309-340
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Robust Single-Walled Carbon Nanotube-Infiltrated Carbon Fiber Electrodes for Structural Supercapacitors: from Reductive Dissolution to High Performance Devices
Advanced Functional Materials, Vol. 33, Núm. 16
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Straightforward Synthesis of Bis[(trifluoromethyl)sulfonyl]ethylated Isocoumarins from 2-Ethynylbenzoates
Journal of Organic Chemistry, Vol. 88, Núm. 11, pp. 7373-7380
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Synthesis of N-Substituted Pyrroles Catalyzed by Low-Cost and Commercially Available Aluminas
Catalysts, Vol. 13, Núm. 3
2022
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1H-imidazo[4,5-f][1,10]phenanthroline carbohydrate conjugates: Synthesis, DNA interactions and cytotoxic activity
Bioorganic Chemistry, Vol. 125
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Graphene-Based Nucleants for Protein Crystallization
Advanced Functional Materials, Vol. 32, Núm. 42
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High- k dielectric screen-printed inks for mechanical energy harvesting devices
Materials Advances, Vol. 3, Núm. 3, pp. 1780-1790