Federico
Gago Badenas
Catedrático/a de Universidad
Instituto de Química Médica
Madrid, EspañaInstituto de Química Médica -ko ikertzaileekin lankidetzan egindako argitalpenak (64)
2023
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Insertion of an Amphipathic Linker in a Tetrapodal Tryptophan Derivative Leads to a Novel and Highly Potent Entry Inhibitor of Enterovirus A71 Clinical Isolates
International Journal of Molecular Sciences, Vol. 24, Núm. 4
2022
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A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro
Pharmaceuticals, Vol. 15, Núm. 8
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Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity
European Journal of Medicinal Chemistry, Vol. 244
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Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library
European Journal of Medicinal Chemistry, Vol. 243
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Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitors
European Journal of Medicinal Chemistry, Vol. 237
2021
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Double Arylation of the Indole Side Chain of Tri- And Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV-1 and EV-A71 Entry Inhibitors
Journal of Medicinal Chemistry, Vol. 64, Núm. 14, pp. 10027-10046
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Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles
Journal of Medicinal Chemistry, Vol. 64, Núm. 9, pp. 6137-6160
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Multivalent Tryptophan- and Tyrosine-Containing [60]Fullerene Hexa-Adducts as Dual HIV and Enterovirus A71 Entry Inhibitors
Chemistry - A European Journal, Vol. 27, Núm. 41, pp. 10700-10710
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Small molecule–peptide conjugates as dimerization inhibitors of leishmania infantum trypanothione disulfide reductase
Pharmaceuticals, Vol. 14, Núm. 7
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The structure and flexibility analysis of the Arabidopsis synaptotagmin 1 reveal the basis of its regulation at membrane contact sites
Life Science Alliance, Vol. 4, Núm. 10
2020
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Hakin-1, a new specific small-molecule inhibitor for the E3 ubiquitin-ligase Hakai, inhibits carcinoma growth and progression
Cancers, Vol. 12, Núm. 5
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N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interaction
European Journal of Medicinal Chemistry, Vol. 194
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Peptides mimicking the β7/β8 loop of HIV'1 reverse transcriptase p51 as “hotspot-targeted” dimerization inhibitors
ACS Medicinal Chemistry Letters, Vol. 11, Núm. 5, pp. 811-817
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Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein–protein interaction disruptor
British Journal of Pharmacology, Vol. 177, Núm. 22, pp. 5163-5176
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Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors
Journal of Medicinal Chemistry, Vol. 63, Núm. 1, pp. 349-368
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Tuning melatonin receptor subtype selectivity in oxadiazolone-based analogues: Discovery of QR2 ligands and NRF2 activators with neurogenic properties
European Journal of Medicinal Chemistry, Vol. 190
2019
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(F)uridylylated peptides linked to VPg1 of foot-and-mouth disease virus (FMDV): Design, synthesis and X-Ray crystallography of the complexes with FMDV RNA-Dependent RNA Polymerase
Molecules, Vol. 24, Núm. 13
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Pyrrolopyrimidine vs Imidazole-Phenyl-Thiazole Scaffolds in Nonpeptidic Dimerization Inhibitors of Leishmania infantum Trypanothione Reductase
ACS Infectious Diseases, Vol. 5, Núm. 6, pp. 873-891
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Structure-Guided Tuning of a Selectivity Switch towards Ribonucleosides in Trypanosoma brucei Purine Nucleoside 2′-Deoxyribosyltransferase
ChemBioChem, Vol. 20, Núm. 24, pp. 2996-3000
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Viral engagement with host receptors blocked by a novel class of tryptophan dendrimers that targets the 5-fold-axis of the enterovirus - A 71 capsid
PLoS Pathogens, Vol. 15, Núm. 5