Isabel
Iriepa Canalda
Profesor/a Titular Universidad
José Luis
Marco Contelles
Publicaciones en las que colabora con José Luis Marco Contelles (48)
2024
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Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors
ACS Chemical Neuroscience, Vol. 15, Núm. 18, pp. 3363-3383
2023
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Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer’s Disease Treatment
International Journal of Molecular Sciences, Vol. 24, Núm. 11
2022
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N-Hydroxy-N-Propargylamide Derivatives of Ferulic Acid: Inhibitors of Cholinesterases and Monoamine Oxidases
Molecules, Vol. 27, Núm. 21
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Polyfunctionalized α-Phenyl-tert-butyl(benzyl)nitrones: Multifunctional Antioxidants for Stroke Treatment
Antioxidants, Vol. 11, Núm. 9
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Synthesis and Antioxidant Properties of HeteroBisNitrones Derived from Benzene Dicarbaldehydes
Antioxidants, Vol. 11, Núm. 8
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The Chemotype of Chromanones as a Privileged Scaffold for Multineurotarget Anti-Alzheimer Agents
ACS Pharmacology and Translational Science, Vol. 5, Núm. 11, pp. 1097-1108
2021
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Privileged quinolylnitrones for the combined therapy of ischemic stroke and alzheimer’s disease
Pharmaceuticals, Vol. 14, Núm. 9
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Studies on the affinity of 6-[(: N -(cyclo)aminoalkyl)oxy]-4 H -chromen-4-ones for sigma 1/2 receptors
RSC Medicinal Chemistry, Vol. 12, Núm. 6, pp. 1000-1004
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Synthesis and Biological Assessment of PyrimidoTacrines as Promising Agents for Alzheimer's Disease Therapy
ChemistrySelect, Vol. 6, Núm. 37, pp. 9975-9980
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Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments
Chemical Record, Vol. 21, Núm. 1, pp. 162-174
2020
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Acetylcholinesterase inhibition of diversely functionalized quinolinones for alzheimer’s disease therapy
International Journal of Molecular Sciences, Vol. 21, Núm. 11, pp. 1-20
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Automated Synthesis of New Quinoxalinetacrines
ChemistrySelect, Vol. 5, Núm. 21, pp. 6491-6493
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Homo-tris-nitrones derived from α-phenyl-n-tert-butylnitrone: Synthesis, neuroprotection and antioxidant properties
International Journal of Molecular Sciences, Vol. 21, Núm. 21, pp. 1-18
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Synthesis of hantzsch adducts as cholinesterases and calcium flux inhibitors, antioxidants and neuroprotectives
International Journal of Molecular Sciences, Vol. 21, Núm. 20, pp. 1-19
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Synthesis, antioxidant properties and neuroprotection of α-phenyl-tert-butylnitrone derived HomoBisNitrones in in vitro and in vivo ischemia models
Scientific Reports, Vol. 10, Núm. 1
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Triazolopyridopyrimidine: A new scaffold for dual-target small molecules for Alzheimer's disease therapy
Molecules, Vol. 25, Núm. 14
2019
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Chromenones as Multineurotargeting Inhibitors of Human Enzymes
ACS Omega, Vol. 4, Núm. 26, pp. 22161-22168
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Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer’s disease therapy
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 34, Núm. 1, pp. 479-489
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Multi-target 1,4-dihydropyridines showing calcium channel blockade and antioxidant capacity for Alzheimer's disease therapy
Bioorganic Chemistry, Vol. 91
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New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H3 Receptor (H3R) Antagonism and Calcium Channels Blockade with Additional Cholinesterase Inhibition
Journal of Medicinal Chemistry, Vol. 62, Núm. 24, pp. 11416-11422