Publications by the researcher in collaboration with Carolina Burgos García (16)

2018

  1. Discovery of potent calpain inhibitors based on the azolo-imidazolidenone scaffold

    European Journal of Medicinal Chemistry, Vol. 157, pp. 946-959

2016

  1. Synthesis of 1-Substituted Isoquinolines by Heterocyclization of TosMIC Derivatives: Total Synthesis of Cassiarin A

    Organic Letters, Vol. 18, Núm. 14, pp. 3378-3381

2015

  1. Isoquinoline Synthesis by Heterocyclization of Tosylmethyl Isocyanide Derivatives: Total Synthesis of Mansouramycin B

    Organic Letters, Vol. 17, Núm. 1, pp. 78-81

2014

  1. Microwave-assisted synthesis of potent PDE7 inhibitors containing a thienopyrimidin-4-amine scaffold

    Organic and Biomolecular Chemistry, Vol. 12, Núm. 24, pp. 4233-4242

2013

  1. Remote aryl cyanation via isocyanide-cyanide rearrangement on tosylmethyl isocyanide derivatives

    Organic Letters, Vol. 15, Núm. 13, pp. 3388-3391

  2. Synthesis and evaluation of quinazoline derivatives as phosphodiesterase 7 inhibitors

    Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 8, pp. 2370-2378

2012

  1. A cascade reaction of azolopyrimidines. Synthesis of unusual indole and azaindole derivatives

    Chemical Communications, Vol. 48, Núm. 73, pp. 9171-9173

2011

  1. Radical intramolecular arylation of pyridinium salts: A straightforward entry to 7-hydroxypyrido[2,1-a]isoquinolinylium salts

    European Journal of Organic Chemistry, pp. 619-628

2010

  1. Application of selective palladium-mediated functionalization of the pyrido[3′,2′:4,5]pyrrolo[1,2-c]pyrimidine heterocyclic system for the total synthesis of variolin B and deoxyvariolin B

    European Journal of Organic Chemistry, pp. 5607-5618

2008

  1. Palladium-mediated C-N, C-C, and C-O functionalization of azolopyrimidines: a new total synthesis of variolin B

    Tetrahedron Letters, Vol. 49, Núm. 25, pp. 4073-4077

2007

  1. Reaction of imines with N-iodosuccinimide (NIS): Unexpected formation of stable 1 : 1 complexes

    Chemical Communications, pp. 1281-1283

  2. Selective palladium-catalyzed amination of the heterocyclic core of variolins

    Tetrahedron Letters, Vol. 48, Núm. 14, pp. 2597-2601

2005

  1. Heterocyclizations with tosylmethyl isocyanide derivatives. A new approach to substituted azolopyrimidines

    Journal of Organic Chemistry, Vol. 70, Núm. 12, pp. 4879-4882

2004

  1. Benzo[f]azino[2,1-a]phthalazinium Cations: Novel DNA Intercalating Chromophores with Antiproliferative Activity

    Journal of Medicinal Chemistry, Vol. 47, Núm. 5, pp. 1136-1148

1999

  1. The first example of an intramolecular Westphal reaction. Synthesis of a new aza-quinolizinium type system

    Tetrahedron Letters, Vol. 40, Núm. 21, pp. 4115-4118

1989

  1. Synthesis and structural, conformational and pharmacological study of N-β(or γ)acyloxyalkylnortropinones

    European Journal of Medicinal Chemistry, Vol. 24, Núm. 2, pp. 123-129