Publicaciones en colaboración con investigadores/as de Eli Lilly and Company (20)

2011

  1. Ethyl 4,4-dimethyl pyroglutamate (DMPG): A chiral auxiliary in cyclopropanation and carbonyl group activator

    Arkivoc, Vol. 2011, Núm. 3

2008

  1. Palladium-mediated C-N, C-C, and C-O functionalization of azolopyrimidines: a new total synthesis of variolin B

    Tetrahedron Letters, Vol. 49, Núm. 25, pp. 4073-4077

2006

  1. Synthesis of L-2-amino-8-oxodecanoic acid: An amino acid component of apicidins

    Synthesis, pp. 2069-2073

2005

  1. Diastereoselective addition of heteroatom nucleophiles to ethyl 2-(diethoxymethyl)cycloprop-2-ene-1-carboxylate

    Arkivoc, Vol. 2005, Núm. 9, pp. 394-404

2003

  1. Chemoselective Nucleophilic Attack on N-Acyl Derivatives of (S)-Ethyl 4,4-Dimethyl Pyroglutamate (DMPG)

    Organic Letters, Vol. 5, Núm. 21, pp. 3791-3794

2002

  1. Unexpected highly regioselective macrocyclization of o-allylic N-carbonyl substituted anilines

    Tetrahedron Letters, Vol. 43, Núm. 45, pp. 8025-8027

1999

  1. A new approach to the synthesis of 2-aminoimidazo[1,2-α]pyridine derivatives through microwave-assisted N-alkylation of 2-halopyridines

    Tetrahedron, Vol. 55, Núm. 8, pp. 2317-2326

  2. Short synthesis and anti-rhinoviral activity of imidazo[1,2- a]pyridines: The effect of acyl groups at 3-position

    Bioorganic and Medicinal Chemistry Letters, Vol. 9, Núm. 10, pp. 1391-1394

1998

  1. New enantioseleetive approach to the total synthesis of (-)-α-Kainic Acid

    Tetrahedron Letters, Vol. 39, Núm. 15, pp. 2171-2174

1997

  1. Stereoselective synthesis of 1,3,4-substituted tetrahydro-β-carbolines from indoles based on selective transformations

    Tetrahedron, Vol. 53, Núm. 24, pp. 8237-8248

  2. Suzuki-type cross-coupling reaction of 1-benzyl-2-iodo-1H-benzimidazoles with aryl boronic acids: A regioselective route to N-alkylated 6-alkoxy-2-aryl-1H-benzimidazoles

    Tetrahedron, Vol. 53, Núm. 37, pp. 12755-12764

1996

  1. 4-Benzyl-2,3-didehydroprolinate as a homochiral template for Michael additions. Synthesis of enantiopure α-allokainoids, β-kainoids, 2,3-methanoprolines and other 3,4-disubstituted prolines

    Tetrahedron Asymmetry, Vol. 7, Núm. 9, pp. 2613-2626

  2. A microwave synthesis of the cis and trans isomers of 3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one : The influence of solvent and power output on the diastereoselectivity

    Tetrahedron Letters, Vol. 37, Núm. 35, pp. 6413-6416

  3. Conformationally constrained serotonin analogues: Stereoselective synthesis of trans -3-(2-aminocycloalkyl)indoles by aziridine ring opening

    Tetrahedron Letters, Vol. 37, Núm. 5, pp. 683-686

  4. Use of azalactones in a 'Pictet-Spengler-like' reaction. Stereoselective synthesis of 1,3,4-substituted tetrahydro-β-carbolines

    Tetrahedron Letters, Vol. 37, Núm. 32, pp. 5813-5816

1994

  1. Diastereoselective functionalization of 5-hydroxy prolinates by tandem Horner-Emmons-Michael reaction

    Tetrahedron Letters, Vol. 35, Núm. 43, pp. 8037-8040

  2. Stereoselective Double Alkylation of Ethyl N-Boc-pyroglutamate

    Journal of Organic Chemistry

1993

  1. General method for the synthesis of 5-arylpyrrole-2-carboxylic acids

    Tetrahedron Letters, Vol. 34, Núm. 39, pp. 6317-6320

1991

  1. New uses of Westphal condensation: Synthesis of flavocorylene and related indolo[2,3-a]quinolizinium salts.

    Tetrahedron Letters, Vol. 32, Núm. 51, pp. 7575-7578

  2. New uses of the westphal condensation. Synthesis of pi-donor-pi-acceptor heterocycles.

    Tetrahedron, Vol. 47, Núm. 35, pp. 7329-7342